Extended knowledge of 1-Methyl-5-nitroimidazole

According to the analysis of related databases, 3034-42-2, the application of this compound in the production field has become more and more popular.

Each compound has different characteristics, and only by selecting the characteristics of the compound suitable for a specific situation can the compound be applied on a large scale. 3034-42-2, name is 1-Methyl-5-nitroimidazole, This compound has unique chemical properties. The synthetic route is as follows., COA of Formula: C4H5N3O2

General procedure: To a solution of 1-methyl-5-nitro-1H-imidazole (10 g, 0.078 mol) in EtOH (400 mL) was added wet10% Pd/C (2 g), and the mixture was stirred at room temperature for 1 hr. Then diethyl 2- (ethoxymethylene)malonate (20 g, 0.094 mol) was added. The mixture was stirred under H2 for overnight. Pd/C was removed after filtration and the solvent was evaporated in vacuum. The residue was purified by flash column (DCM/MeOH = 10/1) to give diethyl 2-(((1-methyl-1H-imidazol-5-yl)amino)methylene)malonate (6 g, yield: 28.7%) as brown oil. MS: m/z 268.1 (M+H).

According to the analysis of related databases, 3034-42-2, the application of this compound in the production field has become more and more popular.

Reference:
Patent; SANFORD-BURNHAM MEDICAL RESEARCH INSTITUTE; PINKERTON, Anthony, B.; HASSIG, Christian, A.; JACKSON, Michael, R.; ARDECKY, Robert, John; PASS, Ian; (436 pag.)WO2016/123392; (2016); A2;,
Imidazole – Wikipedia,
Imidazole | C3H4N2 – PubChem